Direct condensation of functionalized sp(3) carbons with formanilides for enamine synthesis using an in situ generated HMDS amide catalyst.
نویسندگان
چکیده
The efficient synthesis of functionalized enamines including β-enaminoesters was effectively accomplished by the direct condensation of functionalized sp(3) carbanions such as acetates with formamides using in situ generated HMDS base from catalytic cesium fluoride and stoichiometric tristrimethylsilylamine.
منابع مشابه
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ورودعنوان ژورنال:
- Chemical communications
دوره 50 49 شماره
صفحات -
تاریخ انتشار 2014